TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 0.0900nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 0.210nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 0.490nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database
Affinity DataKi: 0.810nMAssay Description:Displacement of [3H]CGP12177 from beta1 adrenergic receptor in rat cerebral cortex by liquid scintillation methodMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database
Affinity DataKi: 2nMAssay Description:Displacement of [3H]CGP12177 from beta1 adrenergic receptor in rat cerebral cortex by liquid scintillation methodMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 2.60nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database
Affinity DataKi: 3nMAssay Description:Displacement of [3H]CGP12177 from beta1 adrenergic receptor in rat cerebral cortex by liquid scintillation methodMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database
Affinity DataKi: 3nMAssay Description:Radioligand receptor binding studies were conducted in the rat brain.More data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 3.40nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database
Affinity DataKi: 4nMAssay Description:Displacement of [3H]CGP12177 from beta1 adrenergic receptor in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 5.10nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database
Affinity DataKi: 5.30nMAssay Description:Compound was evaluated for its Beta-1 adrenergic receptor binding affinity by measuring the displacement of [3H]-dihydroalprenolol binding in rat hea...More data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 5.30nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database
Affinity DataKi: 5.40nMAssay Description:Displacement of [3H]-CGP-12177 from adrenergic beta1 receptor in Wistar rat cortex incubated for 60 mins by microbeta liquid scintillation counting a...More data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 5.80nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 6.5nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 6.60nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database
Affinity DataKi: 7nMAssay Description:Displacement of [3H]CGP-12177 from beta1 adrenergic receptor in rat brain cerebral cortex after 60 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database
Affinity DataKi: 11nMAssay Description:Displacement of [3H]-CGP-12177 from adrenergic beta1 receptor in Wistar rat cortex incubated for 60 mins by microbeta liquid scintillation counting a...More data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database
Affinity DataKi: 11nMAssay Description:Displacement of [3H]CGP12177 from beta1 adrenergic receptor in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database
Affinity DataKi: 15nMAssay Description:Displacement of [3H]-CGP-12177 from beta1-adrenergic receptor in rat brain cortex after 1 hr by Microbeta scintillation counting methodMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database
Affinity DataKi: 20nMAssay Description:Compound was evaluated for its Beta-1 adrenergic receptor binding affinity by measuring the displacement of [3H]-dihydroalprenolol binding in rat hea...More data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 29nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database
Affinity DataKi: 47nMAssay Description:Displacement of [3H]CGP12177 from beta1 adrenergic receptor in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 49nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 49nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database
Affinity DataKi: 51nMAssay Description:Binding affinity against beta1-adrenergic receptor in rat brainMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database
Affinity DataKi: 51nMAssay Description:Binding affinity to rat brain membrane adrenergic beta-1 receptorMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database
Affinity DataKi: 60nMAssay Description:Compound was evaluated for the inhibition of binding of [3H]-dihydroalprenolol from beta-1 adrenergic receptor of rat cerebral cortical membranesMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database